Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10712 |
CCR2 antagonist 3
AZD-2927,AZD2927 |
CCR | Immunology/Inflammation; Microbiology/Virology |
CCR2 antagonist 3 (AZD-2927) 是 CCR2的拮抗剂。 | |||
T35772 |
Emestrin
|
||
Emestrin is a mycotoxin originally isolated from E. striata that has antimicrobial, immunomodulatory, and cytotoxic activities.1,2,3,4,5 It is active against the fungi C. albicans and C. neoformans, as well as the bacteria E. coli, S. aureus, and methicillin-resistant S. aureus (MRSA; IC50s = 3.94, 0.6, 2.21, 4.55, and 2.21 μg/ml, respectively).2 Emestrin is a chemokine (C-C motif) receptor 2 (CCR2) antagonist (IC50 = 5.4 μM in a radioligand binding assay using isolated human monocytes).3 Emestr... |